structure name | K. PNEUMONIAE TOPOISOMERASE IV (PARE-PARC) IN COMPLEX WITH DNA AND COMPOUND 34 (7-[(1S,5R)-1-AMINO-3-AZABICYCLO[3.1.0]HEXAN-3-YL]-4- (AMINOMETHYL)-1-CYCLOPROPYL-3,6-DIFLUORO-8-METHYLQUINOLIN-2(1H)-ONE) |
reference | Bellamacina et al. J.Med.Chem. 63 7773 2020 |
source | KLEBSIELLA PNEUMONIAE 342 |
experiment | X-ray (resolution=3.20, R-factor=?) |
structural superfamily | Type II DNA topoisomerase; |
reference complex | 6waa_D |
links to other resources | NAKB PDIdb DNAproDB |
protein sequence | |
interface signature | KYRSAEIR/KKSAERIR |
Estimated binding specificities ?
readout + contact |
A | 0 0 3 92 11 3 24 24 24 88 0 84 0 96 96 6 C | 0 0 6 0 5 15 24 24 24 0 0 3 96 0 0 84 G | 0 96 3 3 15 65 24 24 24 5 0 3 0 0 0 3 T | 96 0 84 1 65 13 24 24 24 3 96 6 0 0 0 3scan! |
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updated Sat Dec 16 20:27:59 2023